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CDK2 inhibitor 73
CAS No. 2079895-42-2
CDK2 inhibitor 73( CDK2-IN-73 | CDK2 IN 73 | CDK2IN73 | CDK2 inhibitor 73 )
Catalog No. M13236 CAS No. 2079895-42-2
A potent, selective CDK2 inhibitor with IC50 of 44 nM for CDK2/cyclin A, displays 2,000-fold selectivity over CDK1/cyclin B (IC50=86 uM).
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 205 | Get Quote |
|
| 10MG | 335 | Get Quote |
|
| 25MG | 566 | Get Quote |
|
| 50MG | 806 | Get Quote |
|
| 100MG | 1098 | Get Quote |
|
| 200MG | Get Quote | Get Quote |
|
| 500MG | Get Quote | Get Quote |
|
| 1G | Get Quote | Get Quote |
|
Biological Information
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Product NameCDK2 inhibitor 73
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NoteResearch use only, not for human use.
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Brief DescriptionA potent, selective CDK2 inhibitor with IC50 of 44 nM for CDK2/cyclin A, displays 2,000-fold selectivity over CDK1/cyclin B (IC50=86 uM).
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DescriptionA potent, selective CDK2 inhibitor with IC50 of 44 nM for CDK2/cyclin A, displays 2,000-fold selectivity over CDK1/cyclin B (IC50=86 uM).
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In Vitro——
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In Vivo——
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SynonymsCDK2-IN-73 | CDK2 IN 73 | CDK2IN73 | CDK2 inhibitor 73
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PathwayAngiogenesis
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TargetCDK
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RecptorCDK
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Research Area——
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Indication——
Chemical Information
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CAS Number2079895-42-2
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Formula Weight442.497
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Molecular FormulaC23H18N6O2S
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Purity>98% (HPLC)
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SolubilityIn Vitro:?DMSO : 20.83 mg/mL (47.07 mM)
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SMILESO=S(C1=CC=C(NC2=NC(C3=CC(C4=CC=CC=C4)=CC=C3)=C5N=CNC5=N2)C=C1)(N)=O
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Chemical Name4-((6-([1,1'-biphenyl]-3-yl)-9H-purin-2-yl)amino) benzenesulfonamide
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Coxon CR, et al. J Med Chem. 2017 Mar 9;60(5):1746-1767.
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